Evidence supporting the use of: Doxylamine succinate
For the health condition: Sleep (restless and disturbed)
Synopsis
Source of validity: Scientific
Rating (out of 5): 4
Doxylamine succinate is an antihistamine commonly used as an over-the-counter sleep aid in products such as Unisom. Its sedative properties stem from its ability to cross the blood-brain barrier and antagonize central histamine H1 receptors, which are involved in the regulation of wakefulness. There is substantial scientific evidence supporting its efficacy in the short-term treatment of insomnia and sleep disturbances. Multiple randomized controlled trials have demonstrated that doxylamine succinate can reduce sleep latency and increase total sleep time compared to placebo. The American Academy of Sleep Medicine and other clinical guidelines acknowledge the short-term use of first-generation antihistamines like doxylamine for occasional insomnia, though they caution against chronic use due to the risk of tolerance, anticholinergic side effects (such as dry mouth, urinary retention, and cognitive impairment), and next-day sedation. While doxylamine succinate is not considered the first-line treatment for chronic insomnia, its use in supporting sleep, particularly for transient or situational sleep disturbances, is backed by both clinical practice and scientific research. However, long-term safety and efficacy data are limited, and non-pharmacological interventions are generally preferred for persistent sleep disturbances.
More about Doxylamine succinate
More about Sleep (restless and disturbed)
Other ingredients used for Sleep (restless and disturbed)
5-Hydroxytryptophan (5-HTP)ashwagandha
calcium
chamomile
GABA (gamma aminobutyric acid)
hops
iron
L-ornithine
L-tryptophan
magnesium
Melatonin
ophiopogon root
vitamin B6
Zinc
catnip
Swertia
lotus seed
Wood betony
5-Methoxytryptamine
Albizia
Baikal Skullcap
Codonopsis
cannabinol
Calea zacatechichi
Capitate Valerian
cowslip
Doxylamine succinate
Ficus religiosa
Griffonia simplicifolia
Gardenia jasminoides
kiwi
lemon balm
Lactucarium
linden
Lactucopicrin
Large-leaved linden
lily
Mistletoe
mandrake
Night jessamine
orchid
Premna
Pentatropis capensis
poppy
Semecarpus anacardium
Tarragon
Takuna
Other health conditions supported by Doxylamine succinate
InsomniaMorning Sickness
Nausea and Vomiting
Sleep (restless and disturbed)